3D structures from the PDB for "Tyrosine-protein kinase ABL1 [201-500,M351T]" AND "BDBM13530"
(Proteins have >= 85% sequence identity and ligands are exact matches)
| Seq Identity | Jmol Display | PDB Title |
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2HYY | >99% | | HUMAN ABL KINASE DOMAIN IN COMPLEX WITH IMATINIB (STI571, GLIVEC) |
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6NPE | >99% | | C-ABL KINASE DOMAIN WITH THE ACTIVATOR(CMPD6), 2-CYANO-N-(4-(3,4- DICHLOROPHENYL)THIAZOL-2-YL)ACETAMIDE |
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6NPV | >99% | | C-ABL KINASE DOMAIN WITH THE ACTIVATOR(CMPD51), N-(1-(3,4- DICHLOROPHENYL)-4-(2-HYDROXYETHYL)-4,5-DIHYDRO-1H-PYRAZOL-3-YL) ISONICOTINAMIDE |
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6NPU | >99% | | C-ABL KINASE DOMAIN WITH THE ACTIVATOR(CMPD29), N-(1-(3,4- DICHLOROPHENYL)-4,5-DIHYDRO-1H-PYRAZOL-3-YL)ACETAMIDE |
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3PYY | >99% | | DISCOVERY AND CHARACTERIZATION OF A CELL-PERMEABLE, SMALL-MOLECULE C- ABL KINASE ACTIVATOR THAT BINDS TO THE MYRISTOYL BINDING SITE |
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7N9G | >99% | | CRYSTAL STRUCTURE OF THE ABL 1B KINASE DOMAIN IN COMPLEX WITH DASATINIB AND IMATINIB |
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3MS9 | >99% | | ABL KINASE IN COMPLEX WITH IMATINIB AND A FRAGMENT (FRAG1) IN THE MYRISTATE POCKET |
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6HD4 | >99% | | ABL1 IN COMPLEX WITH COMPOUND 7 AND IMATINIB (STI-571) |
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6HD6 | >99% | | ABL1 IN COMPLEX WITH COMPOUND6 AND IMATINIB (STI-571) |
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1IEP | >99% | | CRYSTAL STRUCTURE OF THE C-ABL KINASE DOMAIN IN COMPLEX WITH STI-571. |
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1OPJ | >99% | | STRUCTURAL BASIS FOR THE AUTO-INHIBITION OF C-ABL TYROSINE KINASE |
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